Pay in 4 interest-free payments of $25.00 Learn more
Ships within 48 hours · Estimated delivery Aug 14 - Aug 19
RS-127445 potently antagonizes 5-HT-evoked formation of inositol phosphates (pKB=9
Formula: C19H28BrNO3
74 (5-HT6)
) produces significant inhibition of passive peritoneal anaphylaxis in guinea-pigs
AR-A 2 12952 RS-127445 potently antagonizes 5-HT-evoked formationAR A 2 is a selective 5 HT1B receptor antagonist, with high affinity to guinea pig cortex 5HT1B 1D and recombinant guinea pig 5 HT1B receptors (Ki=0. 24 and 0. 47 nM) and with 10 fold lower affinity to guinea pig 5 HT1D receptor (Ki, 5 nM), and shows an EC50 of 4. 5 nM for the guinea pig 5 HT1B receptor; AR A 2 can be used in the research of depression and anxiety. Product information CAS Number: 220051 79 6 Molecular Weight: 448. 60 Formula: